Table 1.
ISIS No. | Target | Sequence | Chemistry |
---|---|---|---|
383266 | Il4R-α | ACCTCAGCAACAACAGCAC | siRNA |
383268 | Il4R-α | GTGAAGGATCTGCTCCCAG | siRNA |
383270 | Il4R-α | CACAGACCTCAGCAACAAC | siRNA |
383273 | Il4R-α | TTCTGGGAAACCTGCCAGC | siRNA |
383275 | Il4R-α | GTTCTCAGGTGACATGCTC | siRNA |
383281 | Il4R-α | TTTATTGACATAAAGCTCC | siRNA |
383281-2MM | Il4R-α | TTTATTGACATAtAGCTgC | siRNA |
383281-4MM | Il4R-α | TTaATTcACATAtAGCTgC | siRNA |
383281-SCR | Il4R-α | agatcTctacgtctataat | siRNA |
459728 | Il4R-α | TAAAGACTTTATTGACATAA | siRNA |
459730 | Il4R-α | GACAAGATAAAGACTTTATT | siRNA |
459732 | Il4R-α | TATTGACATAAAGCTCCATG | siRNA |
451522 | Il4R-α | TTTATTGACATAAAGCTCC | siRNA |
455185 | Il4R-α | TTTATTGACATAAAGCTCC | siRNA |
29589 | PTEN | TTAAATTTGGCGGTGTCA | siRNA |
29592 | PTEN | TGTCTCTGGTCCTTACTT | siRNA |
29593 | PTEN | ACATAGCGCCTCTGACTG | siRNA |
29600 | PTEN | TGCTAGCCTCTGGATTTG | siRNA |
29604 | PTEN | GTGTCAAAACCCTGTGGA | siRNA |
371864 | Eg5 | CAACAAGGATGAAGTCTAT | siRNA |
549896 | WAF1 | TTTATTGAGCACCAGCTTTG | siRNA |
549894 | GATA3 | TTTAATAAATACCATCAAAA | siRNA |
549900 | STAT2 | TTTATTATGACGTACGAAGG | siRNA |
308299 | Exosc9 | TGCCAAACCTTTTCACCAGC | RNaseH |
454373 | SKIV2l | GCCAGCCTCATCCACATAGC | RNaseH |
395392 | Ago1 | CTGGACTATTTGCATAGCAA | RNaseH |
399560 | Ago3 | GTTTGCCCATAGTGCCATAC | RNaseH |
395927 | Ago4 | GGCTAACAGTCGAATTGGTT | RNaseH |
368473 | Dcp1a | CACCATGTTGCTCAGGGAGG | RNaseH |
365128 | DCP2 | CTGCATGTAGAAATCCAAGT | RNaseH |
443335 | GW182 | TCCTCAGTAGATTTCCATCC | RNaseH |
339800 | DDX6 | CTCGGGTAAACAGATCAGTG | RNaseH |
All siRNA are full RNA in both sense and antisense strand except underlined bases which indicate 2′-O-methoxyethyl substitutions (2′MOE). All RNaseH-dependent ASOs are full phosphorothioate with 2′-O-methoxyethyl substitutions at the positions indicated by underline. Nucleotide mismatches are represented by lower case.