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. 2000 Aug 8;97(17):9363–9364. doi: 10.1073/pnas.180314297

Table 1.

The distribution and ligand affinitives of cannabinoid receptors

Receptor
CB1 CB2
Ligand activity
 Δ9-THC Agonist Weak antagonist
 Cannabidiol Does not bind Does not bind
 Anandamide Agonist Agonist
Tissue distribution
 Greatest activity Brain Immune system