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. Author manuscript; available in PMC: 2012 Jul 24.
Published in final edited form as: J Biomol Screen. 2009 Jun 25;14(7):824–837. doi: 10.1177/1087057109338517

Table 1.

Summary of HTS campaign for screening TNAP using luminescent assay

Compounds screened Hits identified Hit criteria Hit rate
Primary HTS 64,394 73 >50% inhibition 0.11%
Single-concentration confirmation 73 55 >50% inhibition 75.3%
Dose-response confirmation 55 53 IC50 < 20 uM 96.4%