Table 2.
Entry | Ar = | yield[b] |
---|---|---|
2a | 91 | |
2b | 92 | |
2c | 90 | |
2d | 83 | |
2e | 88 | |
2f | 91 | |
2g | 94 | |
2h | 91 | |
2j | 81 | |
2k | 89 |
Conducted at 55–60 °C using 1.5 equiv. LiN(SiMe3)2, 1.5 equiv. ArBr, 3–5 mol % PdCl2(PPh3)2, and THF as solvent
Isolated yields.
Entry | Ar = | yield[b] |
---|---|---|
2a | 91 | |
2b | 92 | |
2c | 90 | |
2d | 83 | |
2e | 88 | |
2f | 91 | |
2g | 94 | |
2h | 91 | |
2j | 81 | |
2k | 89 |
Conducted at 55–60 °C using 1.5 equiv. LiN(SiMe3)2, 1.5 equiv. ArBr, 3–5 mol % PdCl2(PPh3)2, and THF as solvent
Isolated yields.