Table 1.
entry | compound | R | yield |
---|---|---|---|
1 | 3a | -Ph | 85% |
2 | 3b | -CH2OH | 76% |
3 | 3c | -CH2OCH3 | 73% |
4 | 3d | -CH2N(CH3)2 | 56% |
5 | 3e | -(CH2)3CN | 68% |
6 | 3f | -CH2N(CH2CH2)O* | 74% |
7 | 3g | -COOCH3 | 52% |
8 | 3h | -4-Cl-Ph | 95% |
9 | 3i | -CH2CH2OH | 70% |
morpholine
entry | compound | R | yield |
---|---|---|---|
1 | 3a | -Ph | 85% |
2 | 3b | -CH2OH | 76% |
3 | 3c | -CH2OCH3 | 73% |
4 | 3d | -CH2N(CH3)2 | 56% |
5 | 3e | -(CH2)3CN | 68% |
6 | 3f | -CH2N(CH2CH2)O* | 74% |
7 | 3g | -COOCH3 | 52% |
8 | 3h | -4-Cl-Ph | 95% |
9 | 3i | -CH2CH2OH | 70% |
morpholine