Table 4.
MK-5172 potencies against GT1 NS3/4a patient isolates in an NS3/4a phenotype assay
NS3/4a sequence | Genotype | EC50 (nM)a |
---|---|---|
Con1 | 1b | 0.9 ± 0.7 |
H77 | 1a | 1.1 ± 0.6 |
ps20 | 1b | 1.8 ± 0.2 |
ps29 | 1a | 0.4 ± 0.3 |
ps30 | 1b | 5.9 ± 1.4 |
ps31 | 1b | 0.3 ± 0.1 |
ps32 | 1b | 0.6 ± 0.3 |
ps33 | 1b | 4.9 ± 0.4 |
ps36 | 1a | 1.1 ± 0.4 |
ps38 | 1a | 2.8 ± 0.7 |
ps40 | 1a | 0.8 ± 0.1 |
ps41 | 1a | 1.4 ± 0.2 |
Values are means and standard deviations.