Table 2.
SEQUENCE | IC50 CDK2/A2(µM) |
Potency ratio |
IC50 CDK4/D1(µM) |
Potency ratio |
---|---|---|---|---|
SAKRRLFG | 3.3 | 2.9 | ||
HAKRRLIF | 1.3 | 1.5 | ||
RRLIpfF | 26 | 20.0 | 250 | 166.7 |
HAKCitRLIF | 18 | 13.8 | 21 | 14.0 |
HAKTRLIF | 50 | 38.5 | 25 | 16.7 |
CitRLIF | 164 | 126.2 | 179 | 119.3 |
SCCP10 | 25 | 19.2 | 8 | 5.3 |
SCCP 5624 | >100 | 60 | 20.7 | |
SAKRNLFGM | 146 | |||
SAKRNLFG | 75 | |||
SAKRALFGM | 68 | |||
PAKRRLFG | 8 | 6.7 | ||
PVKRRLFG | 3 | 28 | ||
PVKRRL3CFG | 1 | 3.2 |