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. 2012 Jun 6;65(8):397–404. doi: 10.1038/ja.2012.43

Table 2. Calculated pharmacokinetic parameters (mean±s.d.) after intraperitoneal administration of ME0177 (1 mg, 55–60 mg kg−1) and ME0192 (0.53 mg, 28–30 mg kg−1).

Pharmacokinetic parameter ME0177 ME0192
t1/2 (h) 0.66±0.08 5.04±1.06
Tmax (h) 0.26±0.15 1.36±0.58
Cmax (μg ml−1) 17.08±5.5 0.24±0.05
AUC 0-inf_obs (μg ml−1 h) 12.80±3.5 2.15±0.27
MRT 0-inf_obs (h) 0.75±0.14 7.39±1.63
Vz/F_obs ((μg)/(μg ml−1)) 80.99±25.6 2046.13±424.28
Cl/F_obs ((μg)/(μg ml−1) h−1) 86.17±29.9 283.12±37.15