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. Author manuscript; available in PMC: 2012 Aug 29.
Published in final edited form as: J Med Chem. 2009 Mar 12;52(5):1450–1458. doi: 10.1021/jm8014525

Figure 5. Comparison of lucPpy and Ultra-Glo luciferase inhibition for a series of quinoline analogs.

Figure 5

Red fits, solid circles and squares are lucPpy, and black fits, open circles and squares are Ultra-Glo luciferase for 8 (squares) or 9 (circles) assayed using KM levels of substrates. Also shown is the activity of these two compounds using Kinase-Glo for 8 (open triangles) and 9 (upside-down open triangles). The inset shows activity in the qHTS for a series of related quinolines in the lucPpy qHTS (solid circles, red-fits) and Kinase-Glo (open circles).