Table 1.
Compound | IC50 (μM) | Cyt25 (μM) |
---|---|---|
INP0149 | 0.9 | 12.5 |
INP0161 | 1.3 | >25 |
INP0341 | 2.3 | >25 |
INP0400 | 7.3 | >25 |
Compounds were assayed against HIV-1US657, a primary R5 isolate, using TZMbl target cells. Percentage inhibition was calculated based on a DMSO control (no compound). IC50 refers to concentration of compound resulting in ≥50% virus inhibition; Cyt25 refers to concentration resulting in ≥25% cytotoxicity of TZMbl cells by propidium iodine staining.