TABLE 1.
Kinase inhibition profile of CTA056
| Kinase | IC50 |
|---|---|
| μM | |
| Itk | 0.1 |
| Btk | 0.4 |
| Etk | 3 |
| Src | 1.2 |
| Yes | >10 |
| Lyn | >10 |
| Axl | >10 |
| Mer | >10 |
| EGFR | >10 |
| Abl | >10 |
| Mkk1 | >10 |
| PDK1 | >10 |
| Akt | >10 |
| Erk1 | >10 |
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