Table 1.
Uptake of 64Cu-DOTA-GU40C4 and 64Cu-DOTA-Pctrl in major organs of interest determined by quantitative PET imaging analysis.
64Cu-DOTA-GU40C4 | 64Cu-DOTA-Pctrl | |||||
---|---|---|---|---|---|---|
|
||||||
1 h | 4 h | 20 h | 1 h | 4 h | 20 h | |
Tumor | * †2.25 ± 0.24 | ‡2.15 ± 0.34 | * §1.90 ± 0.18 | 0.34 ± 0.12 | 0.30 ± 0.14 | 0.51 ± 0.19 |
Salivary glands | †3.17 ± 0.25 | ‡3.00 ± 0.36 | §1.83 ± 0.21 | 0.28 ± 0.08 | 0.22 ± 0.04 | 0.42 ± 0.10 |
Heart | 1.30 ± 0.27 | 1.50 ± 0.20 | 1.30 ± 0.26 | 0.31 ± 0.11 | 0.32 ± 0.05 | 0.65 ± 0.04 |
Lung | 2.03 ± 0.32 | 1.77 ± 0.31 | 1.33 ± 0.06 | 0.32 ± 0.11 | 0.42 ± 0.13 | 0.52 ± 0.01 |
Liver | 24.03 ± 0.90 | 24.40 ± 0.78 | 18.53 ± 1.31 | 13.57 ± 1.38 | 12.27 ± 1.67 | 11.63 ± 1.56 |
Kidney | 6.57 ± 1.34 | 6.50 ± 1.23 | 5.07 ± 0.91 | 43.47 ± 4.35 | 41.53 ± 3.07 | 30.43 ± 5.66 |
Muscle | 0.49 ± 0.07 | 0.37 ± 0.06 | 0.26 ± 0.02 | 0.14 ± 0.03 | 0.12 ± 0.04 | 0.12 ± 0.03 |
Data are presented as %ID/g ±standard deviation (n = 3).
p = 0.06;
p = 0.004;
p = 0.02;
p = 0.65.