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. 2012 Jun 13;4(9):1345–1352. doi: 10.1002/cctc.201200155

Table 2.

Substrate scope of the pyridine directed direct arylation of compounds 11.Inline graphic

Entry[a] Substrate Boronic acid Product Yield [%]
1 Inline graphic Inline graphic Inline graphic 69
2 Inline graphic Inline graphic Inline graphic 63
3 Inline graphic Inline graphic Inline graphic 65
4 Inline graphic Inline graphic Inline graphic 62
5 Inline graphic Inline graphic Inline graphic 74
6 Inline graphic Inline graphic Inline graphic 83
7 Inline graphic Inline graphic Inline graphic 76
8 Inline graphic Inline graphic Inline graphic 88
9 Inline graphic Inline graphic Inline graphic 57
10 Inline graphic Inline graphic Inline graphic 77
11 Inline graphic Inline graphic Inline graphic 63
12 Inline graphic Inline graphic Inline graphic 57
13 Inline graphic Inline graphic Inline graphic 45
14 Inline graphic Inline graphic Inline graphic 43
15 Inline graphic Inline graphic Inline graphic 50[a]

[a] Bisarylated product 13 formed as a byproduct.