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. 2012 Oct;25(4):682–707. doi: 10.1128/CMR.05035-11

Table 7.

Experimental antimicrobial agents active against carbapenemase-producing Enterobacteriaceae

Drug Compound type Relevant target Reference
BAL30072 Siderophore-containing sulfactam Enterobacteriaceae, including MβL producers 194
Plazomicin (ACHN-490) Sisomicin derivative Gram-negative organisms, including carbapenemase producers 149
GSK2251052 Leucyl-tRNA synthetase inhibitor Gram-negative organisms, including carbapenemase producers 5