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. Author manuscript; available in PMC: 2012 Dec 22.
Published in final edited form as: Bioorg Med Chem Lett. 2011 Sep 28;22(4):1822–1826. doi: 10.1016/j.bmcl.2011.09.047

Table 3.

SAR of the phenethylamine portion

graphic file with name nihms428332t8.jpg
Compd R IC50 (µM)a Selectivityb
BJeLR BJeH-LT
1a graphic file with name nihms428332t9.jpg 0.025 0.578 23
1o graphic file with name nihms428332t10.jpg 0.113 0.27 2.4
1p graphic file with name nihms428332t11.jpg 0.075 0.179 2.4
1q graphic file with name nihms428332t12.jpg 0.089 0.208 2.3
1r graphic file with name nihms428332t13.jpg 0.102 0.242 2.4
a

Values are means of experiments performed in triplicate.

b

BJeH-LT IC50/BJeLR IC50.