TABLE 5.
Results of the inhibition experiments with PBP 2xR
| Inhibitor | Residual activity (%) in presence of inhibitor at concn (μM)a
|
|
|---|---|---|
| 100 | 10 | |
| Arylalkylidene rhodanines | ||
| 2 | 10 | 60 |
| 4 | 20 | 100 |
| Arylalkylidene iminothiazolidin-4-ones | ||
| 7 | 80 | 100 |
| 9 | 10 | 80 |
| 13 | 10 | 60 |
The absolute error was 15% for the competition experiment with PBP 2xR.