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. 2012 Dec 14;55(24):10948–10957. doi: 10.1021/jm301328h

Table 1. Evaluation of 5′-α and β-Thymidine Derivatives against PfTMPK, P. falciparum and MRC5 Cellsc.

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a

hTMPK Ki > 1000 μM.16

b

hTMPK Ki = 362 μM.16

c

Reference compound: chloroquine EC50 = 0.007 μM.