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GSK319197A potencies and affinities
Reporter gene assay and competition binding data are means ± S.E. (n = 2–5).
| HEK-GPR55 | HEK-CB1 | HEK-GPR55+CB1 | |
|---|---|---|---|
| NFAT activation (EC50 in μm) | 0.033 ± 0.013 | ||
| SRE induction (EC50 in μm) | 0.269 ± 0.048 | ||
| Competition binding (Ki in μm) | |||
| SR141716A | 0.4927 ± 0.2555 | 0.0048 ± 0.0012 | 0.0022 ± 0.0001 |
| GSK319197A | 0.2428 ± 0.0494 | 6.2630 ± 4.1452 |
