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. Author manuscript; available in PMC: 2013 Jan 3.
Published in final edited form as: Isr J Chem. 2010 Dec 7;50(5-6):577–587. doi: 10.1002/ijch.201000036

Scheme 21.

Scheme 21

Sequential Larock indole synthesis/cross-coupling.[xlviii] OAc = acetate, S-Phos = 2-dicyclohexylphosphino-2',6'-dimethoxybiphenyl, RuPhos = 2-dicyclohexylphosphino-2',6'-diisopropoxybiphenyl.