Table 2.
Effect of Amino Acid Substitutions in the V2 Region of HIV-1 Env on Ability of HIV-1 V2 mAbs to Bind. See Also Table S4.
mAb | EC50, ug/ml
|
|||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
A244 gp120 | AE.703359 gp120 | AE.427299 gp120 | gp70 B.CaseA2 V1–V2 | |||||||||
WT | K169V | Mut3 | WT | Q169K | Mut3 | WT | Q169K | Mut4 | WT | V169K | Mut3 | |
RV144V2 antibodies: | ||||||||||||
CH58 | 0.03 | 0.05 | 7 | 0.38 | 0.04 | 0.07 | 22.5 | 3.4 | 0.03 | 1.2 | 0.025 | 0.03 |
CH59 | 0.029 | 0.58 | NB | NB | 1.2 | 0.05 | NB | NB | 0.03 | NB | NB | 0.02 |
Other V1V2 antibodies: | ||||||||||||
697D | 0.1 | 0.06 | 0.08 | 0.21 | 0.51 | 0.12 | 0.07 | 0.13 | NB | 0.04 | 0.14 | 0.04 |
PG9 | 0.6 | 3 | >100 | >5 | 0.53 | 0.54 | 0.47 | 0.13 | >10 | NB | >100 | >10 |
PG16 | >10 | >100 | NB | NB | >10 | >10 | >10 | 0.26 | NB | NB | NB | NB |
CH01 | 0.35 | 0.13 | 0.93 | NB | NB | NB | >10 | >10 | NB | NB | NB | NB |
The indicated HIV-1 Env willdtype (WT), and Env mutants with a single a.a residue substitution at the position 169, 3 a. a. residue substitutions (Mut3) or 4 a. a. residue substitutions (Mut4) were assayed in ELISA.
AE.A244 gp120/Mut 3 = K169V/V172E/H173Y.
AE.703359 gp120/Mut 3 = Q169K/R170Q/Q173H.
AE.427299 gp120/Mut 4 = R168K/Q169K//Y173H/A174V.
gp70 B.CaseA2 V1–V2/Mut3 = V169K/E172V/E173H.