. Author manuscript; available in PMC: 2013 Feb 13.

Published in final edited form as: Curr Drug Metab. 2012 Nov;13(9):1345–1355. doi: 10.2174/138920012803341339

Table 1.

Drugs using active transport ^29,30

Transporter	Drugs
Lipid/ Bile Acid Transporters	Fatty acids, lipophilic drugs (?)
Organic Anionic Transporters	Salycilic acid, Statins (e.g. simvastatin, atorvastatin), NSAIDs, fluoroquinolones
Organic Cationic transporters	Dopamine, Verapamil, Cimetidine, Famotidine, Biguanides
Nucleoside Transporter	Antivirals and anticancer compounds
Intestinal Dipeptide Transporter	B-lactams, ACEI^®, thrombin inhibitors
Aminoacid Transporters	Gabapenti, baclofen
Vitamin Transporters	Valproic acid, salicylic acid, methotrexate
P-glycoprotein	Vincristine, paclitaxel, cyclosporin, ciprofloxacin, vinblastine

^®

ACEI Angiotensin converting enzyme inhibitors.