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. 2012 Dec 20;168(2):458–470. doi: 10.1111/j.1476-5381.2012.02145.x

Table 3.

Monoamine release from monoamine-preloaded cells

DAT SERT
EC50 (μM) (95% CI) EC50 (μM) (95% CI)
MDMA 22 (8.9–53) 5.63 (3.5–9.2)
MBDB >100 2.49 (1.0–6.9)
MDEA >100 2.88 (1.6–5.0)
Ethylone >100 9.90 (2.4–40)
Mephedrone 3.75 (1.7–8.4) 5.98 (3.2–11)
Naphyrone >100 >100
Butylone >100 5.5 (1.8–17)
Cocaine >100 >100
Methylone >100 >10
Flephedrone 12.5 (5.7–28) >33
Cathinone 5.64 (3.0–10) >100
Methcathinone 2.36 (1.7–3.3) >33
Amphetamine 1.76 (1.1–2.9) >33
Methamphetamine 1.56 (0.9–2.8) >33
Pyrovalerone >100 >100
MDPV >100 >100

Values are means.