. Author manuscript; available in PMC: 2013 Jul 18.

Published in final edited form as: J Am Chem Soc. 2012 Jul 3;134(28):11350–11353. doi: 10.1021/ja303443m

Table 1.

ortho-Borylation of N-(Boc)-Anilines^a

graphic file with name nihms-391221-t0010.jpg

entry	yield	entry	yield
1	92%^b	7	95%
2	78%	8	82%
3	79%	9	44%
4	89%	10	62%
5	68% ^c	11	40%
6	70% ^d	12	51%

See supporting information for details on conditions. Yields refer to isolated material except as noted

Yield determined by ¹H NMR

Yield is for the major isomer

Isolated as a 92:8 mixture.