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. 2013 Mar 13;8(3):e58485. doi: 10.1371/journal.pone.0058485

Table 1. Selectivity of Tripolins against a panel of kinases.

IC50 values (µM)
Kinase analyzed Tripolin A Tripolin B
Aurora A 1.5 2.5
Aurora B 7.0 6.0
EGFR 11.0 71.7
FGFR 33.4 38.0
KDR 17.9 6.5
IGF1R 14.9 13.2

IC50 values of Tripolin A and Tripolin B against Aurora A, Aurora B and a panel of other selected kinases.