Fig.5. Effects of specific EP receptor antagonists on PGE2 mediated HPSC functions.
HPSC were plated and allowed to settle overnight. Serum containing media was re-plated with serum free media for 24 hours before addition of EP1, EP2 or EP4 antagonists at a dose of 10μM. 1 hour after the antagonist addition, cell migration and invasion were assessed by counting the number of DAPI stained cells that penetrated the migration membrane after 24 h following PGE2 (100nM) stimulation. (A) membrane alone (right, stained cells; left migration numbers p<0.05 versus control) (B) matrigel coated membrane (right, stained cells; left migration numbers p<0.05 versus control). Addition of EP4 antagonist showed a significant reduction of PGE2 mediated HPSC migration and invasion. (C) RT-PCR showing the reduction in collagen 1A1 expression on treatment with EP4 antagonist (10μM) as compared to increase on treatment with PGE2 (100nM) alone.