Table 5.
Thermodynamic Parameters for Binding of LSD1 to CoREST286–482 at Different pH (25 °C) e
| pH | Kd (nM) | ΔH (kcal mol−1) | TΔS (kcal mol−1) | ΔG (kcal mol−1) | Stoichiometry |
|---|---|---|---|---|---|
| 6.0 | 4.18 ± 0.96 | −8.56 ± 0.01 | 2.87 ± 0.66 | −11.4 ± 2.62 | 0.90 ± 0.004 |
| 7.0 | 6.75 ± 1.49 | −12.9 ± 0.15 | −1.54 ± 0.34 | −11.4 ± 2.51 | 1.00 ± 0.01 |
| 8.0 | 7.66 ± 2.91 | −15.6 ± 0.32 | −4.48 ± 1.71 | −11.1 ± 4.22 | 1.00 ± 0.01 |
| 9.0 | nb | nb | nb | nb | nb |
50 mM sodium phosphate, 50 mM glycine, and 1 mM DTT, pH 6.0, 50 mM sodium phosphate, 50 mM glycine, and 1 mM DTT, pH 7.0, 40 mM sodium phosphate, 30 mM glycine, and 1 mM DTT, pH 8.0, 40 mM sodium phosphate, 30 mM glycine, and 1 mM DTT, pH 9.0. nb = no binding curve observed