Table 2.
Hits from general selectivity testing
Target | % inhibition at 10 μM | pIC50 (μM) |
---|---|---|
Aldose reductase (rat) | 98% | 7.4 |
Steroid 5α-reductase (rat) | 88% | 5.2 |
Hits from general selectivity testing
Target | % inhibition at 10 μM | pIC50 (μM) |
---|---|---|
Aldose reductase (rat) | 98% | 7.4 |
Steroid 5α-reductase (rat) | 88% | 5.2 |