Table 2. General in vitro and in vivo features of chCE7agl-[(DOTA)n-decalysine]2 (n = 1, 3, 5).
chCE7agl-[(DOTA)-decalysine]2 | chCE7agl-[(DOTA)3-decalysine]2 | chCE7agl-[(DOTA)5-decalysine]2 | |
Total number of DOTA | 2 | 6 | 10 |
Specific activity | Ca. 70 MBq/mg | Ca. 400 MBq/mg | Ca. 700 MBq/mg |
pI | >9.5 | >9.5 | 7.8–8.3 |
Immunoreactivity | 81.3% | 51.0% | 39.2% |
Tumor-to-blood* | 70.2±24.6 | 15.3±2.2 | 7.9±0.0 |
Tumor-to-Liver* | 1.7±0.9 | 2.2±0.6 | 8.6±0.8 |
Liver-to-blood* | 43.0±7.6 | 7.2±1.2 | 0.93±0.1 |
72 h p.i.