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SAR at N-1.
| |||
|---|---|---|---|
| Compound | R | KD (nM) | |
| BasE | MbtA | ||
| 15 |
|
36.1 ± 4.9 | (3.74 ± 0.41).103 |
| 29 |
|
>100•103 | >100•103 |
| 30 |
|
>100•103 | >100•103 |
| 31 |
|
>100•103 | >100•103 |
| 32 |
|
556 ± 66 | >100•103 |
| 33 |
|
>100•103 | >100•103 |
| 34 |
|
>500•103 | >500•103 |
| 35 |
|
>500•103 | >500•103 |
| 36 |
|
>100•103 | >100•103 |
