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. Author manuscript; available in PMC: 2014 Feb 1.
Published in final edited form as: Bioorg Med Chem Lett. 2012 Dec 20;23(3):614–619. doi: 10.1016/j.bmcl.2012.12.030

Table 2.

NPBWR1 antagonist activity of compounds 9a–9k (IC50 μM)

Compound IC50 (μM)a
9a 0.37
9b 0.49
9c >25
9d 0.53
9e 2.20
9f 3.10
9g 18.00
9h 0.12
9i 0.78
9j 0.43
9k 0.28
a

Data are reported as mean of n = 3 determinations.