Table 2.
F876 mutation frequency in drug-resistant LNCaP/AR xenograft tumors
Treatment | Frequency (%) | Mutation | Endogenous or exogenous locus |
Enzalutamide | 1.06 | F876L | Exogenous |
Enzalutamide | 1.82 | F876L | Exogenous |
Enzalutamide | 2.19 | F876I | Exogenous |
ARN-509 | 1.10 | F876L | Exogenous |
ARN-509 | 1.39 | F876L | Exogenous |
ARN-509 | 71.23 | F876L | Endogenous |