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. Author manuscript; available in PMC: 2013 Apr 12.
Published in final edited form as: Recent Pat CNS Drug Discov. 2012 Dec;7(3):218–229. doi: 10.2174/157488912803252023

Table 1.

Recent patents in Nrf2-ARE pathway activators for treatment of central nervous system disorders.

S.No Patent Application Number Title Applicant PubDate
1 WO/2011/156889 PCT/CA2011/000649 NOVEL MODULATORS OF NRF2 AND USES THEREOF TRT Pharma Inc. 12/22/11
2 WO/2010/107733 PCT/US2010/027394 TREATMENT OF NUCLEAR FACTOR (ERYTHROID-
DERIVED 2)-LIKE 2 (NRF2) RELATED DISEASES BY
INHIBITION OF NATURAL ANTISENSE TRANSCRIPT
TO NRF2
OPKO CURNA,
LLC.
9/23/10
3 WO/2010/036711 PCT/US2009/058050 METHODS OF MODULATING PROTEIN
HOMEOSTASIS, METABOLIC SYNDROME, HEAVY
METAL INTOXICATION AND NRF2 TRANSCRIPTION
FACTORS
Bach Pharma Inc. 4/1/10
4 WO/2009/036204 PCT/US2008/076064 PHASE II DETOXIFICATION AND ANTIOXIDANT
ACTIVITY
Joslin Diabetes center
Inc.
3/19/09
5 WO/2008/136838 PCT/US2007/071933 NOVEL AMIDE DERIVATIVES OF CDDO AND
METHODS OF USE THEREOF
Trustees of
Dartmouth College
11/13/08
6 WO/2008/108825 PCT/US2007/021748 NEUROPROTECTIVE COMPOSITIONS AND METHODS Burnham Institute for
medical research
9/12/08
7 WO/2007/008652 PCT/US2006/026503 METHODS AND COMPOSITIONS DIRECTED TO DJ-1
AS REGULATOR OF THE ANTI-OXIDANT
TRANSCRIPTION FACTOR NRF2
the University of
North Carolina at
Chapel Hill
1/18/07
8 WO/2007/005879 PCT/US2006/026056 COMPOSITIONS AND METHODS FOR THE
TREATMENT OR PREVENTION OF DISORDERS
RELATING TO OXIDATIVE STRESS
The Johns Hopkins
University
1/11/07
9 WO/2008/097596 PCT/US2008/001602 NRF2 SCREENING ASSAYS AND RELATED METHODS
AND COMPOSITIONS
Biogen Idec Inc. 8/14/08