Table 2.
Measurement of biological activity of the released inhibitors, using an enzyme linked sorbent assay. The results were expressed as a percentage activity of TG compared to positive control (without the inhibitor). Results denote mean ±SD from 3 independently synthesized batches.
| % activity of TG |
% reduction in activity of TG |
|||
|---|---|---|---|---|
| Inhibitor (w/w) | 1 % | 0.5 % | 1 % | 0.5 % |
| time | ||||
|
| ||||
| 1 Day | 9.12 | 16.06 | 90.88 | 83.94 |
| 1 week | 6.55 | 12.06 | 93.45 | 87.94 |
| 2 week | 54.34 | 57.90 | 45.66 | 42.10 |
| 3 week | 46.16 | 50.23 | 53.84 | 49.77 |
| 4 week | 78.30 | 82.20 | 21.70 | 17.80 |