Table 1.
TMX in combination with ML141 in vivo suppresses BLBC cell growth
| Normalized photon flux | |||||
|---|---|---|---|---|---|
| 0–50 | 50–100 | 100–150 | 150–200 | 200–250 | |
| Day 0 | |||||
| Ctrl | 6/6 | – | – | – | – |
| TMX | 5/5 | – | – | – | – |
| ML141 | 5/5 | – | – | – | – |
| TMX + ML141 | 6/6 | – | – | – | – |
| Day 7 | |||||
| Ctrl | 5/6 | 1/6 | – | – | – |
| TMX | 5/6 | 1/5 | – | – | – |
| ML141 | 5/6 | 1/5 | – | – | – |
| TMX + ML141 | 6/6 | – | – | – | – |
| Day 14 | |||||
| Ctrl | 1/6 | 3/6 | 1/6 | 1/6 | – |
| TMX | 2/5 | 1/5 | – | 1/5 | 1/5 |
| ML141 | 1/5 | 1/5 | – | 2/5 | 1/5 |
| TMX + ML141 | 5/6 | – | 1/6 | – | – |
Animals were transplanted with 1,000,000 cells and treated with TMX, ML141 or the combination for 14 days. Tumour progression was monitored by whole mouse imaging every 7 days till completion of drug treatment.