Figure 7. Antibodies against p55TNFR protect against TNF toxicity, increase MTD, and allow safe anticancer therapy.
(A) TNF (30 mg) was administered to mice pretreated i.p. with different doses of anti-mp55TNFR monoclonal antibodies (10 mg/ml, n = 5; 5 mg/ml, n = 5; 2.5 mg/ml, n = 4) or PBS (n = 7) or control hamster IgG1 (10 mg/ml, n = 5). (B) Antitumor effects and (C) survival in antitumor experiments on Tnfrsf1a+/+ mice treated for 10 days paralesionally with TNF (25 mg) plus IFN-γ (5,000 IU) (black symbols) or PBS (white symbols) and cotreated i.p. daily with PBS (black), control (red), or anti-mp55TNFR antibodies (gray). (D) Toxicity study of TNF/IFN-γ in B16BL6 melanoma-bearing Tnfrsf1a+/+ mice cotreated i.p. with PBS, control antibodies, or anti-mp55TNFR antibody for 10 days. (E) Human TNFRSF1A knockin mice treated i.p. with anti-hp55TNFR monoclonal antibodies (10 mg/ml, n = 6 or 4 mg/ml, n = 6) or control antibody (10 mg/ml, n = 6) and injected with 50 mg TNF or PBS (n = 6). (F) Antitumor effects and (G) survival in antitumor experiments in human TNFRSF1A knockin mice treated with PBS (white symbols) or TNF/IFN-γ (black symbols) and daily i.p. coadministration of PBS (n = 6), control (n = 6), or anti-hp55TNFR antibodies (n = 12). (H) Toxicity study of TNF/IFN-γ in B16BL6 melanoma-bearing human TNFRSF1A knockin mice i.p. cotreated with PBS, control antibody, or anti hp55TNFR antibody. The horizontal line in D and H represents LD50. In the TSI graphs, “***” is between PBS and TNF/IFN-γ–treated p55TNFR antibody groups. All data represent mean ± SEM. *P < 0.05, **P < 0.01, ***P < 0.001 (Student’s t test in B and F and log-rank test in A, C, E, and G).
