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. Author manuscript; available in PMC: 2013 Jun 3.
Published in final edited form as: Annu Rev Pharmacol Toxicol. 2011;51:267–288. doi: 10.1146/annurev.pharmtox.010909.105812

Table 1.

Mediators released by classically (M1) and alternatively (M2) activated macrophages implicated in liver and lung injury and repair

M1 mediators Toxicant
Liver Lung

Reactive oxygen species Endotoxin (17, 18) Ozone (5961, 63, 64, 101)
Acetaminophen (6, 13, 104) Radiation (65)
Phenobarbital (15) Bleomycin (66)
Carbon tetrachloride (97, 98) Silica (84)
1,2-Dichlorobenzene (100)

Reactive nitrogen species Endotoxin (47, 184) Ozone (59, 6164, 101)
Acetaminophen (12, 25, 44) Radiation (65, 112)
Carbon tetrachloride (40) Bleomycin (66, 111, 113)
Ethanol (114) Silica (115)

Proteases Endotoxin (118) Bleomycin (93)
Acetaminophen (37, 44) Endotoxin (78)
Carbon tetrachloride (134) Sulfur mustard (69, 121)
Thioacetamide (120) Particulate matter (117)

Bioactive lipids Endotoxin (47, 136, 140) Ozone (59, 64, 131, 138, 145)
Acetaminophen (127, 128) Silica (124, 125)
Carbon tetrachloride (97, 126, 130, 134, 148) Sulfur mustard (69)

Proinflammatory cytokines (TNFα, IL-1β, chemokines) Endotoxin (47) Ozone (60, 63, 64, 68)
Acetaminophen (3, 6, 37, 38, 44, 127) Radiation (162)
Carbon tetrachloride (14, 40, 43, 126, 158) Silica (85)
Galactosamine (153) Particulate matter (113, 176)
Cadmium (154) Endotoxin (78)
Asbestos (155, 156)

M2 mediators
IL-10 Endotoxin (47) Ozone (63, 64)
Acetaminophen (37, 38, 44, 49, 50) Silica (91)
Carbon tetrachloride (51) Endotoxin (178)

IL-4 Acetaminophen (38) Radiation (87)
Concanavalin-A (42) Silica (89)
Endotoxin (178)
Hyperoxia (177)

IL-13 Endotoxin (45) Endotoxin (178)
Acetaminophen (46) Hyperoxia (177)
Diesel exhaust (176)

TGFβ Endotoxin (185) Bleomycin (179)
Acetaminophen (38) Radiation (180)
Carbon tetrachloride (43, 126, 182) Asbestos (186)
Thioacetamide (181)

Abbreviations: IL, interleukin; TGFβ, transforming growth factor β; TNFα, tumor necrosis factor α.