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. Author manuscript; available in PMC: 2014 Feb 28.
Published in final edited form as: J Med Chem. 2013 Feb 18;56(4):1739–1747. doi: 10.1021/jm301847z

Table 1.

AlphaScreen IC50 for 3 – 32 (values in µM)

Compound Alpha Compound Alpha
3 > 5 18 NA
4 NA 19 0.18
5 ND 20 NA
6 0.33 21 0.46
7 NA 22 2.8
8 2 23 2.1
9 >10 24 NA
10 0.5 25 ND
11 NA 26 0.76
12 ND 27 0.17
13 ND 28 0.09
14 ND 29 0.43
15 ND 30 2
16 NA 31 0.12
17 NA 32 0.1

ND – compound disrupts the control. NA – no activity at the highest concentration tested.