Table 4. Ligand affinity (IC50) toward GCRPRs.
IC50 [nM] | |||
peptides | chGCRPR | xeGCRPR | mdGCRPR |
GCRP | 43.55±11.11 | 65.53±20.44 | 327.34±51.02 |
chGLP1 | >1000 | >1000 | ND |
huGCG | >1000 | >1000 | ND |
Exe-4 | 217.77±93.19 | 374.11±84.88 | 337.29±42.82 |
Results are presented as mean ± S.E. of at least three independent experiments. ND, not determined.