Table 1.
Substrate hydrolysis by FAAH and MGL enzymes with standard deviations.
Compound | Name | Substrate Assay (% Hydrolysis) | |
---|---|---|---|
FAAH | MGL | ||
1 | 2-AG | 100±0 | 74±4 |
(±)-5 | AM5501 | 91±1 | 48±3 |
(±)-6 | AM5502 | 100±0 | 8±3 |
meso-7 | AM5504 | 2±3 | 2±2 |
(±)-8 | AM5503 | 100±0 | 1±1 |
(+)-8 | AM4434 | 88±2 | 10±3 |
(-)-8 | AM4435 | 88±3 | 13±2 |
meso-9 | AM5505 | 78±6 | 19±4 |