Table 2.
Reactive center loop (RCL) sequences for inhibitory human serpins and generated vaspin variants from residue P15 to P4′
| RCL | |||
|---|---|---|---|
| (P15-----------P1– | -P1'–P4') | ||
| SerpinA1 | Antitrypsin | GTEAAGAMFLEAIPM– | –SIPP |
| SerpinA1variant | Pittsburgh | GTEAAGAMFLEAIPR– | –SIPP |
| SerpinA4 | Kallistatin | GTEAAAATTFAIKFF– | –SAQT |
| SerpinA12 | Vaspin | GTEGAAGTGAQTLPM– | –ETPL |
| SerpinC1 | Antithrombin | GSEAAASTAVVIAGR– | –SLNP |
| SerpinE1 | PAI–I | GTVASSSTAVIVSAR– | –MAPE |
| SerpinA12 variants | VaspinA369P | GTEGAPGTGAQTLPM– | –ETPL |
| VaspinT365R | GREGAAGTGAQTLPM– | –ETPL | |