Table 3. Biochemical and cellular activity of SKII.
IC50 of SKII | |
hSPHK1 (biochemical) [µM] | 17.5 |
hSPHK2 (biochemical) [µM] | 13.0 |
mSPHK1 (biochemical) [µM] | >10 |
mSPHK2 (biochemical) [µM] | >10 |
Endogenous S1P production (LOX) [µM] | 7.5 |
Viability (LOX cells) [µM] | 11.3 |