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. 2011 Jun 27;4(3):210–218. doi: 10.1111/j.1752-8062.2011.00272.x

Table 2.

Expression of BA receptors that regulate cardiovascular function.

BA receptors Tissue type Direct BA action demonstrated References
Nuclear receptors
 FXR Endothelial cells Yes 17, 72
Vascular smooth muscle cells Yes 74, 75, 76
Cardiomyocytes No 17
 PXR Mesenteric arteries No 24
 VDR Cardiomyocytes No 49
G‐Protein‐coupled Receptors
 TGR5 Hepatic sinusoidal endothelial cells Yes 33
Cardiomyocytes No 34
 M2R Cardiomyocytes Yes 30
 M3R Endothelial cells Yes 66
Potassium channels
 BKCa Vascular smooth muscle cells Yes 36, 63