Table 1.
IC50 of Core 1-based analogues (3a–e) against LYP.
![]() | ||
|---|---|---|
| Compd # | IC50 (µM) | |
| 3a | 8.4 ± 0.3 | |
| 3b | 1.82 ± 0.06 |
|
| 3c | 10.0 ± 1 | |
| 3d | 4.2 ± 0.6 | |
| 3e | ![]() |
5.2 ± 0.2 |
IC50 of Core 1-based analogues (3a–e) against LYP.
![]() | ||
|---|---|---|
| Compd # | IC50 (µM) | |
| 3a | 8.4 ± 0.3 | |
| 3b | 1.82 ± 0.06 |
|
| 3c | 10.0 ± 1 | |
| 3d | 4.2 ± 0.6 | |
| 3e | ![]() |
5.2 ± 0.2 |