Table 1.
IC50 of Core 1-based analogues (3a–e) against LYP.
![]() | ||
---|---|---|
Compd # | ![]() |
IC50 (µM) |
3a | ![]() |
8.4 ± 0.3 |
3b | ![]() |
1.82 ± 0.06 |
3c | ![]() |
10.0 ± 1 |
3d | ![]() |
4.2 ± 0.6 |
3e | ![]() |
5.2 ± 0.2 |
IC50 of Core 1-based analogues (3a–e) against LYP.
![]() | ||
---|---|---|
Compd # | ![]() |
IC50 (µM) |
3a | ![]() |
8.4 ± 0.3 |
3b | ![]() |
1.82 ± 0.06 |
3c | ![]() |
10.0 ± 1 |
3d | ![]() |
4.2 ± 0.6 |
3e | ![]() |
5.2 ± 0.2 |