Table 1. IC50 Values of Prodrugs in MCF-7 and T47D Cells.
IC 50 (μM) |
||
---|---|---|
drug | MCF-7 | T47D |
tamoxifen | 0.794 | 1.13 |
4-OHtamoxifen | 0.0291 | 0.210 |
boron prodrug (4) | 0.148 | 0.144 |
boron prodrug (5) | 0.00626 | 0.260 |
boron prodrug (6) | 0.0420 | 0.228 |
IC 50 (μM) |
||
---|---|---|
drug | MCF-7 | T47D |
tamoxifen | 0.794 | 1.13 |
4-OHtamoxifen | 0.0291 | 0.210 |
boron prodrug (4) | 0.148 | 0.144 |
boron prodrug (5) | 0.00626 | 0.260 |
boron prodrug (6) | 0.0420 | 0.228 |