Table 2.
entry | substrate | nucleophile | product | yield (%) |
---|---|---|---|---|
1 |
1 |
22 |
23 |
63 dr = 1:0 |
2 |
1 |
24 |
25 |
71 dr = 1.6:1 |
3 |
1 |
26 |
27 |
65 |
4 |
1 |
28 |
29 |
66 |
5 |
1 |
30 |
– | – |
6 |
14 |
30 |
31 |
46 |
entry | substrate | nucleophile | product | yield (%) |
---|---|---|---|---|
1 |
1 |
22 |
23 |
63 dr = 1:0 |
2 |
1 |
24 |
25 |
71 dr = 1.6:1 |
3 |
1 |
26 |
27 |
65 |
4 |
1 |
28 |
29 |
66 |
5 |
1 |
30 |
– | – |
6 |
14 |
30 |
31 |
46 |