Skip to main content
. Author manuscript; available in PMC: 2013 Dec 1.
Published in final edited form as: Bioorg Med Chem Lett. 2012 Oct 2;22(23):7084–7086. doi: 10.1016/j.bmcl.2012.09.093

Table 2.

IC50 values of SAHA and the C6-SAHA t-butyl variant 2c for HDAC1, HDAC3, and HDAC6

Compound IC50/µM
HDAC1 HDAC3 HDAC6
SAHA 0.096 ± 0.02 0.136 ± 0.01 0.074 ± 0.009
2c 0.99 ± 0.06 5.4 ± 0.7 2.4 ± 0.5