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. Author manuscript; available in PMC: 2013 Aug 22.
Published in final edited form as: J Comb Chem. 2008 Aug 1;10(5):658–663. doi: 10.1021/cc800055x

Table 1.

Library Data for Compounds 6{1–13}

graphic file with name nihms-489942-t0009.jpg

compound R yielda (%) purityb (%)
6{1} 2-ethylphthalimide 40 94
6{2} 2-pyridinyl 30 97
6{3} 1-amino-1-cyclohexyl 42 95
6{4} 4-H2NC6H4 62 99
6{5} 1-methyl-1H-imidazo-5-yl 83 95
6{6} CH2OH 67 97
6{7} 1-hydroxy-1-cyclohexyl 59 99
6{8} 3-thiophenyl 75 97
6{9} 2-(N-methyl)propyl 50 97
6{10} 4-AcOC6H4 60 94
6{11} 4-H2NC6H4 67 93
6{12} 3-O2NC6H4 73 95
6{13} 4-HO2CC6H4 8 87
a

Isolated yield after preparative HPLC.

b

UV purities determined at 214 nm after preparative HPLC.