Table 2.

Library Data for Compounds 6{14–43}

compound	Ar	yielda(%)	purityb(%)
6{14}	5-indolyl	24	92
6{15}	6-methoxy-3-pyridinyl	29	95
6{16}	4-EtO2C-3-FC6H4	53	96
6{17}		5	87
6{18}	6-(N,N-dimethyl)-3-pyridinyl	22	94
6{19}	4-MeO-3-FC6H4	58	97
6{20}	3-MeO2-C-5-O2NC6H4	44	97
6{21}	5-indolyl	51	92
6{22}	6-methoxy-3-pyridinyl	26	95
6{23]	4-EtO2C-3-FC6H4	26	97
6{24}		0
6{25]	6-(N,N-dimethyl)-3-pyridinyl	7	100
6{26}	4-MeO-3-FC6H4	46	88
6{27}	3-MeO2C-5-O2NC6H4	0
6{28}	5-indolyl	79	97
6{29}	6-methoxy-3-pyridinyl	81	95
5{30}	4-EtO2C-3-FC6H4	73	99
6{31}		57	94
6{32}	6-(N,N-dimethyl)-3-pyridinyl	85	96
6{33}	4-MeO-3-FC6H4	73	99
6{34}	3,4,5-(MeO)3C6H4	73	99
6{35}	5-indolyl	75	96
6{36}	6-methoxy-3-pyridinyl	16	91
6{37}	4-EtO2C-3-FC6H4	64	98
6{38}		7	100
6{39}	6-(N,N-dimethyl)-3-pyridinyl	20	92
6{40}	4-MeO-3-FC6H4	60	99
6{41}	3-EtO2C-5-O2NC6H4	0
6{42}	3,4,5-(MeO)3C6H4	53	99
6{43}	3,4-(OCH2CH2O)C6H3	44	99

^aIsolated yield after preparative HPLC.

^bUV purities determined at 214 nm after preparative HPLC.