TABLE 5.
nAChR | IC50 values for PeIA(N11R) | 95% C.I. | IC50 values for PeIA(A7V,S9H,V10A,N11R,E14A) | 95% C.I. |
---|---|---|---|---|
rα3β2 | 30.9 μm | 22.8–42.1 | 35.6 μm | 25.0–50.1 |
rα3K152E,E184D,Q195Tβ2 | 4.07 μm | 3.05–5.44 | 18.2 nm | 15.3–21.7 |
rα6/α3β2β3 | 46.5 nm | 35.0–61.2 | 2.16 nm | 1.98–2.35 |
rα6E152K/α3β2β3 | 1.53 μm | 0.360–6.49 | 311 nm | 215–450 |
rα6E152K,D184E,T195Q/α3β2β3 | 6.20 μm | 0.234–164 | 5.47 μm | 3.20–9.36 |