Skip to main content
. Author manuscript; available in PMC: 2014 Aug 1.
Published in final edited form as: Bioorg Med Chem Lett. 2013 May 29;23(15):4398–4403. doi: 10.1016/j.bmcl.2013.05.072

Figure 3.

Figure 3

Inhibition of Yes1 kinase in a biochemical assay for saracatinib (A, IC50 = 6.2 nM), AMG-Tie-2-1 (B, IC50 = 8.7 nM), AZ-23 (C, IC50 = 39.1 nM).